Lecozotan HCl ( —— )

产品货号. M34311 CAS No. 433282-68-9

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Lecozotan HCl
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Lecozotan HCl (SRA-333) is a potent and selective 5-HT antagonist that significantly enhances KCl-stimulated glutamate and acetylcholine release from the hippocampal dentate gyrus and has cognitive enhancing properties. Chronic administration of Lecozotan HCl did not induce 5-HT(1A) receptor tolerance or desensitization in a behavioral model demonstrating 5-HT(1A) receptor function.
产品描述

Lecozotan HCl (SRA-333) is a potent and selective 5-HT antagonist that significantly enhances KCl-stimulated glutamate and acetylcholine release from the hippocampal dentate gyrus and has cognitive enhancing properties. Chronic administration of Lecozotan HCl did not induce 5-HT(1A) receptor tolerance or desensitization in a behavioral model demonstrating 5-HT(1A) receptor function.
体外实验

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体内实验

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同义词

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通路

GPCR/G Protein
靶点

5-HT Receptor
受体

5-HT Receptor
研究领域

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适应症

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CAS Number

433282-68-9
分子量

520.02
分子式

C28H30ClN5O3
纯度

>98% (HPLC)
溶解度

——
SMILES

[C@H](CN(C(=O)C1=CC=C(C#N)C=C1)C2=CC=CC=N2)(C)N3CCN(C4=C5C(=CC=C4)OCCO5)CC3.Cl
化学全称

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计算器

产品手册

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